Chemistry Services for Drug Discovery

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Special Feature:

Boronic Acids

Chiral Compounds

Functional Groups

Fused Rings

Kinase Inhibitors

Substructure

Name, Cat No, CAS, MDL, etc.

No terms returns ALL

Key Morpholines for the preparation of pharmacologically active compounds.

Morpholine is a common structural feature in drug molecules with varied pharmacological activity: norepinephrine reuptake inhibitors for the treatment of ADHD - WO2005047272 (Lilly); KCNQ family potassium ion channel openers for the treatment of epilepsy - US20100063033 (Lundbeck); leptin receptor modulator mimetics for the treatment of weight gain, type2 diabetes and dyslipidemia – WO2009071678 (AstraZeneca); PI3K kinase inhibitors with multiple potential therapeutic utility - US201000298310 (UCB).

We have launched a comprehensive range of morpholine synthons which are stereochemically defined to facilitate further controlled elaboration.

To view the complete list of our Morpholine synthons, accurate availability and pricing information, please check by substructure search "Morpholine".

2-Substituted Morpholines

(S)-N-Boc-2-Hydroxymethylmorpholine 95+% ee
(R)-N-Boc-2-Hydroxymethylmorpholine 95+% ee
(S)-N-Boc-2-Morpholinecarbaldehyde 95+% ee
(R)-N-Boc-2-Morpholinecarbaldehyde 95+% ee
(R)-N-Boc-2-Morpholinecarboxylic acid 95+% ee
(S)-N-Boc-2-Morpholinecarboxylic acid 95+% ee
(S)-Morpholine-2-carboxylic acid HCl 95+% ee
(R)-Morpholine-2-carboxylic acid HCl 95+% ee
Ethyl Morpholine-2-carboxylate 97%
2-Morpholinecarboxylic acid HCl 97%
2-(Aminomethyl)morpholine 95%
4-Benzyl-2-(chloromethyl)morpholine Hydrochloride 97%

3-Substituted Morpholines

(R)-4-Boc-3-Hydroxymethylmorpholine 95+% ee
(S)-N-Boc-3-Hydroxymethylmorpholine 95+% ee
N-Boc-3-Morpholinecarbaldehyde 95+%
(R)-N-Boc-3-Morpholinecarbaldehyde 95+% ee
(S)-N-Boc-3-Morpholinecarbaldehyde 95+% ee
(S)-N-Boc-morpholine-3-carboxylic acid 95+% ee
(R)-N-Boc-Morpholine-3-carboxylic acid 95+% ee
Methyl 3-Morpholinecarboxylate 97%
4-Boc-3-Morpholinecarboxylic Acid 97%
(S)-Morpholine-3-carboxylic acid 95+% ee
(R)-Morpholine-3-carboxylic acid 95+% ee
3-Morpholinecarboxylic acid 95+%
3-Benzylmorpholine HCl 95+%
(R)-3-Methylmorpholine HCl H2O 95+% ee
3,3-Dimethylmorpholine 95+%
(R)-Morpholin-3-ylmethanol HCl 95+% ee
3-Morpholinemethanol 95+%
Morpholine-3-carbonitrile 95+%
(R)-3-(Methoxymethyl)morpholine HCl 95+% ee
(S)-3-(Methoxymethyl)morpholine HCl 95+% ee
3-(Methoxymethyl)morpholine 95+%

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Chemistry Services for Drug Discovery