Chemistry Services for Drug Discovery

www.activate-scientific.com

MSDS-COA

Activate Scientific GmbH
Am Mitterweg 12
83209 Prien, Germany
Tel: +49 [0] 8051 / 965 16 60
Fax: +49 [0] 8051 / 965 16 61
info@activate-scientific.com

21A The Maltings, Roydon Road
Stanstead Abbotts, Hertfordshire SG12 8HG, UK
Tel: +44 [0] 1279 / 84 32 44

Special Feature:

Boronic Acids

Chiral Compounds

Functional Groups

Fused Rings

Kinase Inhibitors

Substructure

Name, Cat No, CAS, MDL, etc.

No terms returns ALL

Series of Synthons

, upon customers´ request, develops Series of Synthons which have the same core structure but various functional groups. Our chemistry expertise is within smaller complex, fused Heterocyclic Ring systems, carrying various substituents and multiple functional groups at diffcult ring positions.

Please call on us for your specific Custom development project.

Examples of developed Series of Synthons, up to 50g quantities

3-Bromo-5,6,7,8-tetrahydro-1,6-naphthyridine HCl 95+%
7-(tert-Butoxycarbonyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine-3-carboxylic acid 95+%
Ethyl 5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine-3-carboxylate HCl 95+%
tert-butyl 5,6-Dihydro-3-methoxy-[1,2,4]triazolo[4,3-a]pyrazine-7(8H)-carboxylate 95+%
2,4-Dichloro-1,8-naphthyridine 95+%
2-Chloro-5,6,7,8-tetrahydro-1,6-naphthyridine HCl 95+%
Ethyl 4-chloro-1,8-naphthyridine-3-carboxylate 95+%
2-Chloro-1,6-naphthyridine 95+%
Ethyl 1,7-naphthyridine-3-carboxylate 95+%
2-Amino-5-formylthiazole 96%
2-Bromo-5-thiazolecarboxylic acid 97%
2-Fluoropyridine-4-boronic acid 97%
2-Fluoropyridine-3-boronic acid 97%
4-Bromo-2-isopropylthiazole 98%
2-Fluoro-5-(tributylstannyl)pyridine 96%

is a fully equipped service provider of Heterocyclic Custom Building Blocks for research projects in preclinical development

  • Series of heterocyclic Synthons, 5-50g
  • Multistep Custom Synthesis, 7-8 steps up to 5-10g
  • Exclusive Blocks ™, 5-10g
  • Heterocyclic Custom chemicals, up to 1-2kg
  • Fine Intermediates, Production of Fine heterocyclic Intermediates for pilot plant development

We provide very competitive pricing.

Custom made compounds are usually delivered within three to four weeks if it is a two- or three-step synthesis and in one kilogram quantity or less. For more information, call us at +49-(0)8051-9657660, or send an email to rschmitt@activate-scientific.com.

Chemistry Services for Drug Discovery